2006 11 26 2007 03 13 2007 11 09 2009 11 16 2011 09 01 2013 01 22 2013 11 07 Ceftriaxone Sodium for Injection Zhusheyong Toubaoqusongna (6R,7R)-7-[[(2--4- )( )]]-8--3-[[(1,2,5,6--2- -5,6- -1,2,4--3- )]]-5--1-[4.2.0] -2- -2- C 18 H 16 N 8 Na 2 O 7 S 3 3 1/2 H 2 O 1 / 12
661.59 C 18 H 18 N 8 O 7 S 3 1.0 g 0.5 g 0.25 g 12 1~2 24 4 12 14 20~50 / 50 / 2kg 15 12 20~80 / 50 50 / 30 2 / 12
48 72 100 4 4 6 7 50 / 2 14 250 30~90 1~2 5-10 / 2 6 2-8 24 0.25 0.5 1% 2 1 3.5 1 3 / 12
0.25 0.5 5 1 10 2~4 30 2 40 0.45%2.5% 5%10%5% 6%6~10% 3.45% 19% 14% <500/mm 3 10 20g 5% 1.4% 1% Stevens Johnson Lyell / 0.27%1.86% 2.77% 1 mm 2g 30 12 mm 48 mg/dl 6 mm 24 mg/dl 4 mm 16 mg/dl - 4 / 12
3 80mg/kg 10g 2-4 28-1 2 cephamycin 5%~10% 20% 3 4 5 CDAD 5 / 12
A B A B CDAD CDAD CDAD CDAD 6 7 8 5ml/ 2 9 10 11 12 13 6 / 12
ALTAST - Y - 6 2~8 24 2kg 7 / 12
B B C β - β- A β-b β-ab 8 / 12
* * *** ** * ** * * * ** * - ** - - - * *- ß- NCCLS 9 / 12
mg/l =8 16 32 =64 30 µg mm =21 20 14 =13 DIN ICS 1 2~3 81 / 100% 7~12 1~2 60 24 24 <100 / 95% 300 / 85% 50~100 24 1.4 / 4 18 / 17% 4% 10 / 12
50 2~24 10~22 / 5~12 / 50~60% 40~50% 8 70%8 75 2~3 20 15 1 / 36 2010 H10983036 H10983037 H10983038 1100 11 / 12
201203 (021)28922888() (021)50801800 www.roche.com.cn Rocephin 12 / 12