... 1 ASPIRIN... 1 ASPIRIN ARGI... 7 ASPIRIN DL LY... 9 METAMIZOLE SODIUM... 10 PHENYLBUTAZONE... 12 BENORI... 14 PARACET... 16 DIFLUNISAL... 18 CARBASALATE CALCIUM... 20 CHOLINE MAGNESIUM TRISALICY... 22 SALSA... 23 MAGNESIUM SALICY... 25 BENZBROMARONE... 25 I
ALLOPURINOL... 27 PROBENECID... 29 SULFINPYRAZONE... 31 ACEMETACIN... 33 PIROXICAM... 34 PIRPROFEN... 36 BENZYDAMINE... 37 IBUPROFEN... 38 BUFEXAMAC... 39 HELICID... 40 FENOPROFEN... 41 FENOPROFEN CALCIUM... 42 FENBUFEN... 43 FLURBIPROFEN... 45 FLUFENAMIC ACID... 46 CLIDANAC... 46 MEFENAMIC ACID... 47 II
MECLOFENAMIC ACID... 52 AURANOFIN... 55 CARPROFEN... 56 CLOFENAMIC ACID... 57 LOXOPROFEN... 57 IMIDAZATE... 58 NABUMETONE... 59 NAPROXEN... 60 SPANTOL... 63 OXYPHENBUTAZONE... 63 SULINDACT... 64 DICLOFENAC... 66 KETOROLAC... 67 KETOPROFEN... 69 TOLMETIN... 70 DULCITOL... 73 EPIRIZOLE... 74 III
ETHENZAMIDE... 75 PROPYPHENAZONE... 75 INDOMETACIN... 76 ALPRAZOLAM... 79 ESTAZOLAM... 81 OXAZEPAM... 83 BACLOFEN... 84 BUTOCTAMLDE SEMISUCCLNATE... 85 BENZOCTAMIN... 86 DIAZEPAM... 87 BROMAZEPAM... 90 BUSPIRONE... 91 OXAZOLAM... 93 CLORAZEPATE DIPOTASSIUM... 94 FLUDIAZEPAM... 95 FLUTAZOLAM... 96 IV
FLUTOPRAZEPAM... 97 FLURAZEPAM... 98 FLUNITRAZEPAM... 101 ORYZANOL... 102 HALAZEPAM... 103 MENROBAMATE... 104 CARISOPRODOL... 105 LORAZENAM... 106 CHLORDIAZEPOXIDE... 107 CBXAZDAM... 109 ETHYL LOFLAZEPATE...110 CHLORMEZANONE...111 CLONAZEPAM...112 MEXAZOLAM...115 HYDROXYZINE...117 NORDAZEPAM...118 TRIAZOLAM... 120 V
NITRAZEPAM... 121 ETIFOXLNE... 122 ETIZOLAM... 123 FLUSPIRILENE... 126 REDEPTIN IMAP... 126 (7C) PERPHENAZINE ENANTHATE 126 (7) FLUPHENAZINE ENANTHATE... 127 FLUPHENAZINE... 127 HALOPERIDOL DECANOATE 129 FLUPENTIXOL DECANOATE... 130 CHNPENTHIXOL DECANOATE.. 130 PIPOTIAZINE PALMITATE... 130 (11C)PIPOTIAZINE UNDECYLENATE... 132 PENNURIDOL... 133 VI
HALOPERIDOL... 134 DROPERIDOL... 137 PIMOZIDETE... 138 TRIFLUPERIDOL... 139 TIMIPERONE... 140 BROMPERIDOL... 143 PERPHENAZINE... 145 FLUPHENAZINE... 146 THIORIDAZINE... 148 CHLORNROMAZINE... 148 PROCHLORPERAZINE... 156 MESORIDAZINE... 156 TRIFLUPROMAZINE... 157 TRIFLUONERAZINE... 158 ACEPROMAZINE... 159 FLUPENTIXOL... 160 CLOPENTHIXLO... 161 VII
CHLORPROTHIXENE... 162 TIOTIXENE... 163 ZUCLOPENTHIXOL... 164 OXYPERTINE... 168 RISPERIDONE... 168 TIAPRIDE... 170 CLOZAPLNE... 173 CLOTIAPINE... 174 MOLINDONET... 175 MOSAPRAMINE... 176 NEMONAPRIDE... 178 TRIMETOZINE... 180 REMOXIPRIDE... 181... 184 SULTOPRIDE... 186 ZOTEPINE... 187 AMITRIPTYLINE... 188 VIII
AMOXAPINE... 191 AINFBUTAMONE... 193 OPIPRAMOL... 194 AMFETAMINE... 194 IX
Aspirin ( Acetylsalicylic Acid) 2 3 50% 90% 90% 10% 3 5 1
(1) (2) (3) ( 12 6 ) (4) ( 90% ) (5) (1) 0.3 0.6g 1 3 (2) 1 0.6 1g 1 3 4g 2
1 3 1 0.1g/kg 3 3 (3) 1 0.3g 0.6g 1 2 (4) 1g 2 3 2 3 24 (5) X 0.6 0.9g 4 (6) 50mg (7) 1 5000 2 4 3
(1) 40 (2) (1 3g ) K( 2 4mg) (3) ( 2/3) (4) (5) (6) 4
5% 0.9% (1 1 2 1 1000 1500ml) ( ) (200mg/kg) K (7) (8) 5
(9) ( ) (10) (11) (12)10 Reye 0.5g 0.05g 0.1g 0.2g 0.3g 0.3g 0.5g 150 250ml 0.3g 0.5g 0.1g 0.3g 0.45g 0.5g 1 0.3 0.6g 1 0.9 1.8g 1 3 1 0.1g 1 1 3 6 1 0.1 0.15g 1 1 6
2 6 1 0.15 0.3g 1 2 1 0.6 1g 1 3 4g ( ) 0.324g 0.0324g 0.0972g 0.0033g 1 3 1 12 243 6 Aspirin argi 7
1g 1 2 10 25mg/kg 0.9% 2 4ml (1) (2) 40 (3) (4)3 0.5g( 0.25g) 1g( 0.5g) 8
Aspirin DL ly ( dl-lysine-acetylsalicylate ASPEGIC Venopirin Aspisol) ph 5 6 36 120 1.8 0.9 1.8g 2 1 10 25mg/kg 4ml 0.9% 9
( ) 0.9g( 0.5g) 0.5g( 0.28g) Metamizole Sodium ( Analgin NOVALGIN) Noramidopyrine ( ) ( ) 10
0.25 0.5g 0.75 1.25g 10% 20% 5 1 2 1 5 0.25 0.5g 5 10mg/kg (1) (2) ( ) (3) (4) (5) 11
(6) 0.5g 8 10mg/kg 0.25g 0.5g 0.25g(1ml) 0.5g(2ml) 10% 20% Phenylbutazone ( BUTAZOLIDIN BUTADION) Vd120ml/kg 12
Vd t 1/2 56 86 (Oxyphenbutazone) (1) 1 0.3 0.6g 3 1 0.8g 1 0.1 0.2g (2) 0.2g 1 3 1.2 3g (1) 10% 20% (2) 13
(3) 1 1 (4) (5) (6) 25mg ( )( ) 0.1g 600mg(3ml) 200mg Benori ( Benasprate Benorylate BENORAL) 14
t 1/2 1 4g 1 2g 1 3 4 1 0.5 1.5g 1 1.5 4.5g 3 1 25mg/kg 1 4 1 2 250mg 1 4 3 5 500mg 1 3 6 12 500mg 1 4 1g 1 3 4 (1) 15
(2) 0.2g 0.5g Paracet ( Acetaminophen) t 1/2 75 180 25% 50% 1 0.3 0.6g 1 0.6 1.8g 1 2g 10 12 16
1.5g/M 2 2 3 160mg 4 5 240mg 6 8 320mg 9 10 400mg 11 480mg 1 0.15 0.25g 4 1 (1) (2) (3) t 1/2 (4)3 0.3g 84mg 0.3g 0.5g 0.5g 17
0.25g(10ml) 0.15g 0.3g 0.6g 1 0.3 0.6g 1 1 2 3 12 1 0.15 0.3g 1 1 0.075g(1ml) 0.25g(2ml) Diflunisal ( DOLOBID) PG 2 3 t 1/2 8 12 90% 18
1 8 12 500mg 650mg 1g 4g 1000mg 8 12 500mg 500 1000mg 1 1500mg (1) 3% 9% (2) (3) 19
(4) (5) (6) (7) 250mg 500mg Carbasalate Calcium ( Carbaspirin Calcium) 1 0.6 1.2g 20
2 4 24 3.6g 61 50mg 61 1 50 100mg 1 4 1 0.1 0.15g 4 6 1 0.15 0.2g 6 9 1 0.2 0.25g 9 14 1 0.25 0.3g 2 4 (1) (2) (3) 0.1g 0.05g 0.6g 0.3g 0.2g 0.15g 21
Choline Magnesium Trisalicy ( ) t 1/2 9 17 (1) (2) 12 1.5g( ) 1 2 22
1g( ) 1 2 293mg 362mg 440mg 544mg Salsa ( Sasapyrin Sali cylsalicyclic Acid Salicyl Sali cylate Salysal) 2 2 10 30mg/dl(12 ) 16 23
1 0.3 3 1 0.9 1.2g 1 2 3 0.6g 1 1 (1) (2) 0.5g (3) 0.3g 0.5g 24
Magnesium Salicy 1 0.5 1g 1 3 250mg 250mg Benzbromarone ( Exurate) 25
24 66.5% 40 80mg 1 3 6 (1) 18 6 ( 54%) 10 ( 38%) 2 89% (2) (3) 26
Allopurinol ( Isopurinol ZYLORIC ZYLOPRIM) 70% (t 1/2 12 30 ) t 1/2 1 3 0.05g 2 3 2 3 0.2 0.4g 2 3 0.1 0.2g 2 3 8mg/kg 0.1 0.2g 1 4 300mg 27 1
(1) (2) 4 8 (3) (4) 6- (6-MP) 6-MP 1/4 (5) C ( ) (6) (7) 28
3 4 0.1g probenecid ( benemid probalan) (1) (2) ( 29
) (1) 0.25g 2 4 1 0.5 1g 2 (2) 0.5g 4 25mg/kg 3 9 1 (1) (2) (3) 30
0.25g Sulfinpyrazone ( ANTURAN) (1) (2) 6 31
(3) t 1/2 3 0.1 0.2g 2 400 800mg 1 100 400mg 2 (1) 2 (2) (3)10% 15% (4) (5) 0.1g 32
Acemetacin 2.6 99% 1 30mg 3 (1) (2) (3) 33
(4) 30mg Piroxicam ( FELDEEN) 198 202 85% 34
20mg 4 7 t 1/2 45 5% 1 20mg 1 40mg 1 4 6 1 10 20mg 1 (1) (2) (3) 35
20mg(2ml) ( ) ( )10mg 20mg Pirprofen PG t 1/2 6 7 99.5% 24 80% 800mg 1 2 600mg 1000mg/3 1 2 200 400mg 1200mg 400mg 36
(1) (2) 200mg Benzydamine ( BENZYRIN) 1 3 1 25 50mg 37
25mg Ibuprofen ( BRUFEN FENBID) 74.5 77.5 38
0.4 0.8g 3 4 0.2 0.4g 4 6 0.3g 0.1g 0.2g Bufexamac ( DROXAROL FEXIMAC) 153 155 0.75g 1.5g 5% 39
5% ( ) 85.14% 50.9% 10 (1) (2) (3) (4) 0.25g(5g) 0.5g(10g) 0.25g Helicid ( ) 40
(Helicid essatia Hook) 75 100mg 3 7 1 25mg Fenoprofen ( NALFON) 300mg 600mg 300mg 41
t1/2 2.5 0.6g 1 3 4 1 1 0.3 0.6g 1 1 4 0.8g 1 4 Fenoprofen Calcium 0.3g 0.6 0.2g 0.3g 0.2g tmax 1h 2h t1/2 3h 99% 90% 24h 42
0.3g 0.6g/ 3 4 / 0.2g/4h 3.2g/ 6h 1 Fenbufen ( LEDERFEN NAPONOL) BUFEMID 185 188 43
87% O 2 t 1/2 12 17 0.6 0.9g 44
0.9g 0.6g (1) 1 (2)14 (3) ( ) ( )150mg Flurbiprofen (Froben) 500mg 100mg 45
1 150 200mg t1/23.5 Flufenamic Acid 0.2g ( ) 1 0.2g 1 3 Clidanac (Britai) 46
PG 30 45mg 2 3 (1) (2) 30 45mg 2 3 15mg Mefenamic Acid ( Penstel) 47
48 2-[(2 3- ) ] C15H15NO2 241.29 0.25g/ 0.25g/ LD50 780mg/kg LD50 630mg/kg tmax 2h 67% 25% t1/2 2h 1g 2 4 10 g/ml 4 2 ( 20 g/ml) T1/2 267% 25%
(l) (2) (3) (4) (5) 49
(6) (7) (8) (9) (10) 0.5g 0.25g/6h 5mg/kg 3 / 1 50
(1) (2) 7 (3) (4) (5) 51
(6) 14 Meclofenamic Acid ( ) (PH8.7) 189 192 52
( ) 0.5 1 t 1/2 2 200 400mg 3 4 1 400mg 53
2 3 (1) (2) (3) (4) (5) 50mg 100mg 54
Auranofin ( RIDAURA) 29% 25% 60% 40% 12 1 6mg 3mg 1 3mg 2 1 /6mg 6 9mg 3 3 55
(1) (2) (3) 3mg 3mg( 0.87mg) 3mg Carprofen ( Imadvl) 150mg 56
1 150mg 1 2 Clofenamic Acid 0.2g ( ) 1 0.2 0.4g 1 3 Loxoprofen 60mg ( ) 57
60mg 3 Imidazate (Selezen) 0.5 1.5g 1 2 6 12 250 500mg 1 3 20 40 1 3 6 12 10 20 500mg 100mg 500 1000mg 5% 58
500mg 750mg 40%(40g/100ml) 500mg(2ml) 100mg 500mg 750mg 5% Nabumetone t 1/2 24 1.0g 59
0.5g Naproxen ( NAPROSYN) PG 1 2 4 99% t 1/2 13 14 95% ( ) 1 7 60
1 0.2 0.3g 1 2 3 0.5 0.75g 0.375 0.75g 2 0.5g 6 8 0.25g 1.25g 1 100 200mg 1 1 1 0.25g 1 0.5g (1) 61
(2) (3) (4) (5) t 1/2 0.1g 0.125g 0.25g 0.125g 0.2g 0.25g 100mg(2ml) 200mg(2ml) 0.25g 62
Spantol 200mg 1 0.2 0.4g 1 3 Oxyphenbutazone 0.1g ( ) 1 0.1 0.2g 1 3 1 0.1 0.2g 63
Sulindact ( Clinoril) Clinoril 0.1g 0.2g 5-90% t1/2 7h 8h t1/2 16h 18h 64
100mg 200mg/ 2 / 7 1 4.5mg/kg 2 6mg/kg 4.5mg 6mg/ B ( D ) 2 ( ) 65
Diclofenac ( VOLTAREN) 282 285 2 2.5 26 50 1 2 25mg 3 50mg 2 75mg 1 66
(1) (2) (3) 25mg 75mg(2ml) 50mg 1% ( CATAFLAM) 25mg 50mg 12.5mg 25mg 75mg 15mg 75mg(3ml) Ketorolac (KETOROL TORADOL TORATEX) PG 24 67
6 8 50% 10mg 1 1 4 20 30mg 1 3 4 30mg 60mg 1 90mg 150mg 6 20 30mg 10 30mg (1) (2) 68
(3) 30mg(1ml) 10mg Ketoprofen ( PROFENID) 93 96 1 0.5 2 t 1/2 1.6 1.9 24 30% 90% 69
50mg 1 150mg 3 4 100mg 1 3 1 2 25mg 50mg Tolmetin ( TOLECTIN) 155 157 ( ) 70
20 60 t 1/2 24 99% 50% 70% (2 ) 12 71
600 1200mg 75 150mg 4.5g 1 400mg 1 3 600 1800mg 1 15 30mg/kg 1 20mg/kg 600mg (1) 1200mg 25% 40% 5 8% (2) 72
(3) (4) (5) (99%) (6) (7) 200mg Dulcitol (Dulcite) (Tripterygium hypoglau cum) 73
188 189 1 100mg 3 3 1 25mg 1 30 1 ( 50mg 2% 6ml) 3 5 5 7 25mg(2ml) 50mg Epirizole ( Mepirizol DA 398 MEBRON) 74
50mg 1 150 450mg 2 4 Ethenzamide ( ) 1 0.05 0.25g 1 1.0 1.5g Propyphenazone 0.15g 1 0.15 0.3g 75
Indometacin ( Indomethacin INTEBEN INDOCIN) 158 162 (PG) (1) (2) (3) Behcet Batter 76
(4) 90% t 1/2 7 12 25mg 1 2 3 ( ) 100 150mg 3 4 1 50mg 1 50 100mg 10 1 1 75mg 1 25mg 2 1 75mg 2 (1) ( ) 77
78 (2) ( ) (20% 50%) (3) ( ) (4) ( ) (5) (6) (7) 25mg 25mg 25mg 25mg 50mg 100mg 25mg 75mg
100mg(10g) 2 3 Alprazolam ( Xanax) 10-1 2-10 12 19 t 1/2 79
80 1 0.4 0.8mg 1 0.8 1.6mg 0.25 0.5mg 3 4mg 0.25mg 2 2 4mg 10mg 0.4 0.8mg 0.25mg 3 (1) (2) (3)
(4) (5) H 2 t 1/2 (6)18 0.25mg 0.4mg 0.5mg 1mg Estazolam ( EURODIN) 229 232 81
2.4 4 1 2mg 2 4mg 6 12mg 2 4mg 1 1 2 1mg 2mg 82
Oxazepam ( Adumbran Serax Serenid) 4 15 30mg 1 2 3 83
15mg 30mg Baclofen ( LIORESAL) GABA - 5mg 10mg 25mg 3 1 5mg 15 20mg (LIORESAL INTRATHECAL) 0.05mg(1ml) 10mg(20ml) 10mg(5ml) 84
Semisucclnate Butoctamlde (Listomin s) 200mg 24 1 200mg 85
( ) ( ) Benzoctamin ( Tacitin) 10mg 2 10 20mg 3 86
Diazepam ( VALIUM Diapam Stesolid Stesolin) 5 - (GABA) (REM) 70% 80% 87
5 10 1 t 1/2 20 50 2.5 5mg 3 15 30mg 88
5 10mg 6 2.5 10mg 2 4 6 0.1mg/kg 3 10 20mg 4 1 (1) (2) (3) ( 3 ) 89
(1) (2) (3) (4) 2.5mg 4mg 10mg(2ml) Bromazepam ( Lectopam,Lexotanil) 90
1.5mp 3mg 6mg 1.5 3mg 3 2 6 12mg 3 2 Buspirone ( Buspar) 0.5 1 5-1-(2- ) 91
( 1-PP) 10mg 2 3 1 20 30mg 40mg 2 2 3 (1) (2) (3) 18 92
(4) 5mg 10mg Oxazolam 185 189 30 60 10 20mg 3 1 2mg/kg (1) 93
(2) (3) (4) (5) MAOI 5mg 10mg 20mg 10mg 10%( ) Clorazepate DiPotassium ( Tranxene) 11.25mg 22.5mg 3.75mg 7.5mg 15mg 94
15mg 30mg 1 15mg Fludiazepam 0.25mg 1mg/g ( 7.5mg ) 95
7.5mg 3 Flutazolam 4mg ( ) 12mg 3 96
ALT AST Flutoprazepam 2mg (Restas) ( ) 2 4mg 97
4mg ALT AST Flurazepam ( Dalmadorm Dalmane Dormodor Felison) (EMG) (EOG) 98
17 7 8 (REM) REM 28 LD 50 870mg/kg 1232mg/kg 568mg/kg 80mg/kg 10mg/kg N 1 - ( 22% 55%) 15 30mg 15mg 15 99
(1) (2) 15mg (3) (4) (5)15 (6) (7) 100
(8) (9) 15mg 30mg Flunitrazepam ( Rohypnol Darkene) 5 7 ( ) 135 1 2 2mg 101
2mg (1) (2) 2mg 2mg Oryzanol ( ) 102
( ) 3 10mg 60mg 3 10mg Halazepam ( Paxipam) 20mg 40mg 5mg 10mg 3-103
20 40mg 3 80 160mg 20mg Menrobamate ( MILTOWN Eguanil) 103 107 2 3 10% t 1/2 10 104
0.2g 3 4 0.2 0.4g 4 6 0.4g 0.2g 0.4g 0.1g Carisoprodol ( RELA) ( ) 0.35g 3 4 105
(1) (2) (3) 0.35g Lorazenam ( Ativan Lorax Quait) 85% t 1/2 10 18 1 2 6mg 2 4 2 4mg 106
1 4mg 0.5mg 1mg 2mg 2mg(2ml) 4mg(2ml) Chlordiazepoxide ( LIBRIUM) ( ) 4 107
20 24 1 5 10mg 1 15 40mg 1 20mg 3 1 5 10mg 5 5mg 1 3 10 20mg 1 10 20mg 1 30 60mg 25 50mg 5mg/kg 2 1 3 4 (1) ( ) 108
(2) (3) ( ( ) (4) (5) 3 3 5mg 10mg 50mg 100mg Cbxazdam ( Enadel Tolestam 1mg 109
3 12mg Ethyl Loflazepate 2mg (Victan) 1.5 t 1/2 77 1 3mg( 2mg) 1 2mg 110
Chlormezanone ( Fenard REXAN Chlormethazanone) 116 118 0.2g 1 3 111
(1) (2) 0.2g Clonazepam ( CLONOPIN) 237 240 5 1 2 112
6 8 t 1/2 22 38 1 0.75 1mg 2 3 1 4 8mg 2 3 10 20 g/kg 2 3 100 200 g/kg 2 3 1 1 2mg 1 2 4mg 1 1 4mg 0.02 0.06mg/kg 20 2 (1) 113
(2) (3) (4) (1 6 ) (5) (6) 1mg(1ml) 0.5mg 2mg 114
Mexazolam ( Melex) - 1 2 115
1.5 3mg 3 1.5mg (1) (2) (3) ALT AST (4) (5) 116
(6) 0.5mg 1mg 0.1% Hydroxyzine ( Atarax Vistaril) 1 3 1 25 50mg 6 117
50 100mg 4 100 200mg (1) (2) (3)6 50mg 200mg(2ml) 25mg Nordazepam (NORDAZ) 118
97% t 1/2 65 7.5mg 15mg 1 3.75mg (1) (2) (3) 3 3 (4) 119
(5) (6) 7.5mg Triazolam ( Clorazolam Halcion) 239 243 45 30 10 0.25 0.5mg 5mg 15 30mg (15 30 ) 90% t 1/2 2.7 120
0.25 0.5mg 0.25mg Nitrazepam ( Mogadon Nitrados Surem) 121
78% 2 t 1/2 1 25 5 10mg 5 15mg 3 200mg (1) (2) (3) 5mg Etifoxlne (Stresam) 150mg 122
150mg 7 30 Etizolam ( DEPAS) 0.1mol/L 123
146 149 3 5 (2 ) t 1/2 3 t 1/2 8 16 124
1 1mg 3 0.5mg 3 1 1 3mg 1.5mg (1) ALT AST (2) (3) 0.5mg 1mg 10mg 125
Fluspirilene 1 2mg(1ml) Redeptin Imap 1 2mg(1ml) (7C) Perphenazine Enanthate 2 126
(7) Fluphenazine Enanthate 2 4 25mg(1ml) Fluphenazine (Prolixin Decanoate) 9 20 42 72 48 96 2 4 127
25mg 2 4 1 (1) (2) 6 (3) (4) 25mg(1ml) 128
Haloperidol Decanoate ( Haldol Decanoate) 9 20 24 72 6 3 4 1 1 1 50 100mg 1 100 200mg 1 250 300mg 50mg(2ml) 100mg(2ml) 129
Flupentixol Decanoate 2 3 20mg(1ml) Chnpenthixol decanoate 3 4 0.2g(1ml) Pipotiazine Palmitate ( ) 130
(Pipotiazin) 50mg 1 50 100mg 3 4 1 50 200mg 8 16 1 131
(1) (2) (3) 50mg(2ml) 100mg(4ml) Undecylenate (11C)Pipotiazine 2 3 132
1000mg(4ml) Pennuridol 105 108 1 7-133
30 40mg 1 120mg (1) (2) (3) 5mg 20mg Haloperidol ( SERENASE) 134
2 3 72 15% (1) 1 4 60mg 1 2mg 135
1 0.5 1.5mm (2) 1 5 10mg 1 2 3 (3) 5mg 25% 1 2 8 1 (1) (2) (3) (4) (5) (6) 136
(7) 5mg(1ml) 2mg 4mg Droperidol ( Dridol Inapsine) ( ) 137
(1) 1 10 30mg 1 2 (2) 5mg 0.1mg 2 3 5 6 1 (3) 2.5 5mg 5mg(1ml) Pimozidete ( Opiram Orap) 2mg 4mg 10mg 138
4 8mg 1 1 20mg Trifluperidol ( TRIPERIDOL) 2 4mg 2.5 10mg 1 3 0.5mg 2.5mg(1ml) 139
Timiperone (Tolopelon) 4 4.4 14 C 140
0.5 3mg 3 12mg (1) ( ST T PQQT ) ALT AST ( ) 141
(2) (3) (4) 142
(5) (6) (7) (8) 0.5mg 1mg 3mg 10%( g 10mg) Bromperidol (Impromen) 143
4 6 20.2 30.0 3 18mg 36mg (1) ALT (2) 144
(3) 1% 1mg 3mg 6mg Perphenazine ( TRTILAFON) 1 6 12mg 145
1 30 60mg 1 5 10mg 1 5mg 5mg(1ml) 2mg 4mg Fluphenazine ( PERMIFIL Prolixin) 1 1 10mg 1 10 30mg 146
(1) ( ) (2) (3) 5mg(2ml) 2mg 5mg 2mg(1ml) 147
Thioridazine ( Thioril Mellaril) 200mg 10mg 25mg 50mg 100mg 50 100mg 3 800mg 30 200mg Chlornromazine ( WINTERMINE 148
Aminazine) 194 198 (1) - 149
(2) (3) ( ) ( 34 ) (4) (5) - ( 150
) (6) ( ) 2 4 6 90% 10 7- t 1/2 6 9 6 151
(1) 1 12.5 50mg 1 50 800mg 25 50mg 2 3 300 450mg 1 100 150mg (2) 1 25 50mg 152
1 25 100mg (3) 5 10mg 1 1 2 0.5mg (1) (2) 1 2 (3) (4) 153
(5) ( ) (6) 1 40mg (7) 154
( ) (8) 1% (9) 5mg 12.5mg 25mg 50mg 10mg(1ml) 25mg(1ml) 50mg(2ml) 2ml 25mg 2ml 50mg 5ml 50mg ( * ) 100mg 5% 250ml * 100mg 50mg 0.6 0.9mg 5% 250ml 3 5g 0.2 0.3g 6g 1500ml 155
Prochlorperazine ( Compazine) 5mg 10mg 25mg 5mg(1ml) 2.5mg 5mg 25mg 50 100mg 5 10mg 3 15 30mg Mesoridazine ( Serentil) 10mg 25mg 50mg 100mg 156
25mg(1ml) 50mg 3 400mg 25mg 30 60 200mg Triflupromazine 10mg(1ml) (VESPRIN) 10mg 25mg 50mg 157
30 150mg Trifluonerazine ( Stelazine Terfluzine) 1 5 10mg 1 15 4mg 30mg 1 1 2mg 1 2 60% 158
1mg 5mg Acepromazine ( PLEGICIL) 10mg 20mg(2ml) 50mg 100mg 20mg 5% 250ml 10mg 2 20mg 0.2mg 20mg( 0.1 159
Flupentixol ( Flunen thixol Hydrochlo ride Fluanxol 0.5mg Depixol) 3mg 4 8 3mg 2 3 9mg 2 1mg 2 3mg 160
3 Clopenthixlo 10mg ( ) 10mg 1 75mg 2 10 40mg 3 161
Chlorprothixene ( TARDAN) (1) 75 200mg 162
400mg 1 90 150mg (2) 5 25mg 1 3 (1) (2) (3) 12.5mg 15mg 25mg 50mg 30mg(1ml) Tiotixene ( Thiothixene NAVANE) 5mg 10mg 4mg(2ml) 163
5mg 2 20 30mg 60mg 4mg 80mg 2 12mg 2 4 Zuclopenthixol (Sedanxol Cisordlnol Clopixol) 20 10 164
3 6 25% t 1/2 20-75 150mg 10 40mg 2mg 2 6mg 10mg 20 70mg 10 40mg 25mg 25 50mg 2 3 75mg 165
25 50mg 20 75mg (20 75 ) 2 40mg(2 40 ) 1 3 (1) (2) (3) 166
6 12 1 (1) (2) (3) 11.83mg( 10mg) 29.58mg( 25mg) 2.38 11.90 29.75mg( 2 10 25mg) 1ml(20 ) 23.8mg 20mg 14.2%(V/V) 1ml 20ml ( ) 29.58mg ( 25mg) 167
Oxypertine ( Equipertine Forit) 40mg 80 120mg 300mg 30 40mg Risperidone ( Risperidal) 5-HT 2 168
D 2 1 t 1/2 24 1mg 2 3 3mg 1 4 6mg 0.5mg 2 1mg 2mg 3mg 4mg 169
Tiapride ( TIAPRIDAL TIAPREDEX) 197 199-1 170
4( 3 ) 31%( ) 18%( ) - ( ) 171
(1) - 150 300mg( 600mg) 3 2 3 150 300mg (2) 24 200 400mg (3) 200 400mg( 300mg) 3 8 200 400mg 3 50mg 1 3 (4) 24 600 1200mg 4 8 1 3 4 150 800mg 150mg 400mg 172
(5) 7 12-50mg 1 2 (1) ( 2.5%) ( ) (2) 100mg(2ml) 100mg Clozaplne ( Leponex) 173
25mg 50mg 1 100 300mg 2 3 25 75mg 150 3O0mg 500 1000mg 100mg (500mg) Clotiapine (Clothiaoin) 40mg 50mg 174
60 120mg 240mg Molindonet ( Lidone Moban) 5mg 10mg 15mg 25mg 50mg 100mg 20mg(2ml) 50 75mg 3 4 100mg 2 4 15 20mg 175
Mosapramine (Clospipramine Cremine) 2 D 2 5-HT 2 6 7 t 1/2 15 30 150mg 3 300mg 176
(1) (2) 18% (3) (4) (5) 10mg 15mg 25mg 10% 177
Nemonapride (Emonapride Emirace) D 2 - - M- 2 3 t 1/2 2.5 4.5 9 36mg 3 60mg 178
(1) (2) (3) (4) (5) 179
(6) (7) 3mg 10mg Trimetozine ( Sedoxazin TRIOXAZINE) 121 180
300mg 3 6 300mg Remoxipride D 2-5-HT NA Ach GABA 2 C max AUC t 1/2 4 7 (71 89 ) t 1/2 2 181
300mg 2 150 450mg 600mg 1 400mg 300mg 1 150 450mg 600mg 1 2 150mg 150mg (1) 182
ALT (2) (3) (4) - 75mg 150mg 300mg - 150mg 300mg - 100mg(1ml) 25mg(1ml) 25mg(1ml) 110mg(1ml) - 183
( DOGMATIL EQUILID) 177 180 (1) 166 142 5 (2) 184
(1) 600 1200mg (2) 1 100 800mg 300 600mg 1 600 1200mg 1 200 600mg 1 300 600mg 4 1 2 (1) (2) (3) 185
(4) (5) (6) (7) (8) 100mg 50mg(2ml) 100mg(2ml) Sultopride ( Barnetyl) 186
100mg 0.4 1.2g 2.4g 0.4 0.6 1.6 1.8g Zotepine ( Lodopin) 25mg 50mg 100mg 10%100mg(1g) 50%500mg(1g) NA DA 5 HT 5-HT 187
1 4 t 1/2 8 75 100mg 450mg ALT AST Amitriptyline ( Amitid Amitril Elavil Tryptizol) 188
195 199 NA 7 10 8 12 90% t 1/2 9 25 3 189
(1) 25mg 2 150 300mg 50 150mg 50mg 1 (2) 10 25mg 1 11 25 50mg (1) (2) (3) 190
(1) 10 14 (2) (3) (4) 10mg 25mg Amoxapine ( Demolox Moxadil Asendin) NA ( 5-HT 191
) 1 2 10 7-8- t 1/2 6.5 30 50mg 3 100mg 600mg (1) 192
(2) 50mg 100mg 150mg Ainfbutamone ( Bupropin Well butrin) 75mg 5-HT NA 225mg 3 450mg MAOI 18 193
Opipramol ( Insldon Ensidon) 50mg 150 300mg 2 3 50mg 2 Amfetamine ( Amphetamine BENZEDRINE Phenamine) 194
1 2 10mg 1 20mg 1 30mg 1 2 1 10mg 1 20mg 10mg (1) (2) (3) 5mg 10mg 195
5mg(1ml) 10mg(1ml) 196